Isentress and Isentress HD (Raltegravir)

Complete patient guide for uses, dosage, side effects, and safety information

Prescription Required

Quick Facts

Generic Name
Raltegravir
Drug Class
Integrase Inhibitor
Used For
Treatment of HIV in adults and children over 2 years old who weigh at least 25 kg.
How Taken
Oral tablet taken twice daily or once daily, depending on the formulation.

What Is Isentress and Isentress HD Used For?

Isentress and Isentress HD are medications used in combination with other anti-HIV treatments to manage HIV infection.

Primary Uses

They are primarily used to treat HIV in adults and children aged 2 years and older who weigh at least 25 kg.

How It Works

Isentress works by blocking HIV integrase, an enzyme essential for HIV replication, thereby reducing the viral load in the blood.

Good to know: Isentress is not addictive.

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How to Take Isentress and Isentress HD

Follow your doctor's instructions on how to take Isentress or Isentress HD for effective treatment.

Dosage Instructions

Adults should take one 400 mg Isentress tablet twice daily or two 600 mg Isentress HD tablets once daily. Children’s dosages will be determined by their doctor based on weight.

What If You Miss a Dose?

If you miss a dose, take it as soon as you remember. If it’s almost time for your next dose, skip the missed dose. Do not take a double dose.

Important: Never double the dose to make up for a missed dose.

Available Tablet Strengths

400mg
400mg Tablet Pink, Oval • 227
600mg
600mg Tablet Yellow, Oval • 242

Side Effects

Like all medications, this medicine can cause side effects. Most are mild and temporary, but some require medical attention.

Common Side Effects

These side effects occur relatively frequently and usually don’t require emergency care:

  • Nausea
  • Headache
  • Diarrhoea
  • Tiredness
  • Inflammation of nasal passages and throat
  • Trouble sleeping
  • Upper respiratory tract infection
  • Cough
  • Fever
  • Bronchitis
  • Back pain
  • Depression

Seek immediate medical attention if you experience:

  • Severe skin reactions
  • Hypersensitivity reactions
  • Frequent infections
  • Abdominal pain
  • Loss of appetite
  • Fainting
  • Fast or irregular heartbeat
  • Wheezing

Important Warnings

It's crucial to understand the warnings associated with Isentress and Isentress HD.

Who Should Not Take Isentress and Isentress HD

Do not take Isentress if you are allergic to raltegravir or any of its ingredients.

Medical Conditions to Discuss

Inform your doctor about any other medical conditions, medications you are taking, or allergies.

Pregnancy and Breastfeeding

Consult your doctor if you are pregnant or planning to become pregnant. Isentress should not be taken during pregnancy unless advised by your doctor. Breastfeeding is not recommended while taking this medication.

Drug Interactions

Certain medications may interact with Isentress, affecting its effectiveness.

  • Atazanavir
  • Antacids
  • Rifampin
  • Tipranavir/Ritonavir
  • Phenytoin
  • Phenobarbitone

Alcohol & Driving

Be cautious when consuming alcohol and operating machinery while on Isentress.

Alcohol

Consult your doctor about alcohol consumption while taking Isentress.

Driving and Operating Machinery

Be careful when driving or using machinery until you know how Isentress affects you.

Storage

Store Isentress in a cool, dry place below 30°C, away from moisture and heat, and out of reach of children.

Overdose Information

If you suspect an overdose, seek medical attention immediately. Contact your doctor or the Poisons Information Centre at 13 11 26.

Frequently Asked Questions

The time it takes for Isentress and Isentress HD to work can vary by individual, but they are designed to help reduce the amount of HIV in the blood.

Isentress can be taken with or without food.

No, Isentress is not considered addictive.

Stopping Isentress suddenly can lead to an increase in the virus in your blood and may cause HIV to become harder to treat.

Consult your doctor regarding alcohol consumption while on Isentress.

Weight gain is not listed as a common side effect of Isentress.

Elderly patients should discuss their overall health and any medications with their doctor before starting Isentress.

If you miss a dose, take it as soon as you remember, but skip it if it's almost time for your next dose.

Important Disclaimer

This information is intended for general educational purposes only and should not be considered medical advice. Always consult your healthcare provider or pharmacist before starting, stopping, or changing any medication.

If you think you may have a medical emergency, call your doctor or emergency services immediately.

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